SCHEMBL5197284

SCHEMBL5197284

CCC(CC=Cc1cnc2occc2c1)NC(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.35
AAK1 Q2M2I8 5/20 0.35
CTSS P25774 4/20 0.35
CTSK P43235 4/20 0.35
LMNA P02545 2/20 0.35
TP53 P04637 2/20 0.35
XBP1 P17861 2/20 0.35
MAPK1 P28482 2/20 0.35
HTT P42858 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HSD17B10 Q99714 2/20 0.35
HPGD P15428 2/20 0.35
JAK2 O60674 1/20 0.35
S1PR4 O95977 1/20 0.35
F2 P00734 1/20 0.35
HSP90AA1 P07900 1/20 0.33
GAA P10253 1/20 0.33
PKM P14618 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224582 0.83 CDK8 (0.36) SYKAAK1JAK2HDAC4HDAC1
SCHEMBL620441 0.77 AAK1 (0.34) AAK1
SCHEMBL620440 0.77 AAK1 (0.34) AAK1
SCHEMBL6462039 0.77 CHRNB2 (0.48) SYKAAK1CTSSCTSKHPGD
SCHEMBL6451899 0.76 SYK (0.38) SYKAAK1CTSKLMNAHPGD
SCHEMBL5197176 0.76 AAK1 (0.40) SYKAAK1CTSSCTSKALDH1A1
SCHEMBL3910417 0.74 CHRNB2 (0.55) SYKAAK1CTSSCTSKHPGD
SCHEMBL5197286 0.72 CA1 (0.35) AAK1CTSSCTSKLMNAHDAC4
SCHEMBL7529058 0.69 SYK (0.40) SYKAAK1CTSSCTSKATM
SCHEMBL14746635 0.67 ATM (0.48) SYKCTSSCTSKHDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814852-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
EP-1814853-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
WO-2006053082-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed
WO-2006053039-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed