SCHEMBL5197286

SCHEMBL5197286

CC(=CCC(C)NC(=O)OC(C)(C)C)c1cnc2occc2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.34
ATM Q13315 1/20 0.34
TRPA1 O75762 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRB2 P47870 1/20 0.34
NTRK1 P04629 1/20 0.34
AAK1 Q2M2I8 7/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC3 O15379 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224591 0.84 CDK8 (0.39) CA1CA2CA4CA7CA9
SCHEMBL6451903 0.76 NNMT (0.41) CA1CA2CA4CA7CA9
SCHEMBL5197178 0.75 CYP1A2 (0.41) LMNAMAPTAAK1
SCHEMBL6462042 0.75 ACACB (0.35) CA1CA2CA4CA7CA9
SCHEMBL3910420 0.73 CHRNB2 (0.38) CA1CA2CA4CA7CA9
SCHEMBL7529061 0.68 CA2 (0.40) CA1CA2CA4CA7CA9
SCHEMBL620440 0.67 AAK1 (0.34) AAK1
SCHEMBL620441 0.67 AAK1 (0.34) AAK1
SCHEMBL5988005 0.67 CTSS (0.41) ATMGABRB1GABRB2CTSSCTSK
SCHEMBL5987163 0.66 CTSS (0.38) MAPTGABRB1GABRB2CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814852-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
EP-1814853-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
WO-2006053082-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed
WO-2006053039-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed