SCHEMBL5200574

SCHEMBL5200574

CS(=O)(=O)Nc1cc(Br)cc(CC2=NCCN2)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 7/20 0.49
HTR1B P28222 6/20 0.49
RAD52 P43351 1/20 0.43
ADRA1A P35348 6/20 0.41
ADRA2A P08913 4/20 0.41
ADRA1D P25100 4/20 0.41
ADRA1B P35368 4/20 0.41
TAAR1 Q96RJ0 3/20 0.41
ADRA2C P18825 3/20 0.41
ADRA2B P18089 2/20 0.41
CYP2D6 P10635 2/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.41
PTGIR P43119 1/20 0.39
NFKB1 P19838 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5202905 0.99 HTR1D (0.48) HTR1DHTR1BRAD52ADRA1AADRA2A
SCHEMBL5204185 0.86 HTR1D (0.49) HTR1DHTR1BRAD52ADRA1AADRA2A
Hydrochloric Acid SCHEMBL5205837 0.85 HTR1D (0.48) HTR1DHTR1BRAD52ADRA1AADRA2A
SCHEMBL5205731 0.83 HTR1B (0.55) HTR1DHTR1BRAD52ADRA1AADRA2A
SCHEMBL5200685 0.81 HTR1B (0.56) HTR1DHTR1BRAD52ADRA1AADRA2A
SCHEMBL4992561 0.80 LMNA (0.58) HTR1DHTR1BRAD52ADRA1AADRA2A
Hydrochloric Acid SCHEMBL5201578 0.80 HTR1B (0.54) HTR1DHTR1BRAD52ADRA1AADRA2A
SCHEMBL5201043 0.78 HTR1D (0.44) HTR1DHTR1BRAD52ADRA1AADRA2A
Hydrochloric Acid SCHEMBL5200632 0.77 HTR1D (0.43) HTR1DHTR1BRAD52ADRA1AADRA2A
SCHEMBL4990044 0.77 HTR1D (0.51) HTR1DHTR1BRAD52ADRA1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed