SCHEMBL5200685

SCHEMBL5200685

CS(=O)(=O)Nc1cccc(CC2=NCCN2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 4/20 0.56
TAAR1 Q96RJ0 5/20 0.52
ADRA1A P35348 4/20 0.52
ADRA2C P18825 3/20 0.52
ADRA1D P25100 3/20 0.52
ADRA1B P35368 3/20 0.52
CYP2D6 P10635 2/20 0.52
ADRA2A P08913 2/20 0.52
ADRA2B P18089 2/20 0.52
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
TSHR P16473 1/20 0.52
PARP1 P09874 1/20 0.50
NFKB1 P19838 1/20 0.49
RAD52 P43351 1/20 0.47
NR3C1 P04150 1/20 0.46
HTR1D P28221 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5201578 0.99 HTR1B (0.54) HTR1BTAAR1ADRA1AADRA2CADRA1D
SCHEMBL4992561 0.84 LMNA (0.58) HTR1BTAAR1ADRA1AADRA2CADRA1D
SCHEMBL5204185 0.82 HTR1D (0.49) HTR1BTAAR1ADRA1AADRA2CADRA1D
SCHEMBL5200574 0.81 HTR1D (0.49) HTR1BTAAR1ADRA1AADRA2CADRA1D
Hydrochloric Acid SCHEMBL5205837 0.81 HTR1D (0.48) HTR1BTAAR1ADRA1AADRA2CADRA1D
Hydrochloric Acid SCHEMBL5202905 0.80 HTR1D (0.48) HTR1BTAAR1ADRA1AADRA2CADRA1D
SCHEMBL5201601 0.79 NISCH (0.56) HTR1BADRA1AADRA2CADRA1DADRA1B
SCHEMBL5205731 0.79 HTR1B (0.55) HTR1BTAAR1ADRA1AADRA2CADRA1D
SCHEMBL5200888 0.79 RAD52 (0.49) HTR1BTAAR1ADRA1AADRA2CADRA1D
SCHEMBL4993472 0.79 RAD52 (0.49) HTR1BTAAR1ADRA1AADRA2CADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed