SCHEMBL5200731

SCHEMBL5200731

CCOc1ccc(NC(=O)Nc2ccc(OC(F)F)cc2)cn1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.59
NPC1 O15118 2/20 0.55
MAPT P10636 7/20 0.52
RAB9A P51151 4/20 0.52
PKM P14618 1/20 0.52
KMT2A Q03164 8/20 0.51
MEN1 O00255 7/20 0.51
PABPC1 P11940 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
LMNA P02545 3/20 0.47
PAX8 Q06710 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
POLB P06746 2/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
MAPK1 P28482 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4119219 0.87 KDM4E (0.77) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL4105198 0.85 MAPT (0.68) KDM4ENPC1MAPTRAB9APKM
SCHEMBL5198659 0.82 KDR (0.51) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL4110390 0.80 MEN1 (0.62) NPC1MAPTRAB9APKMKMT2A
SCHEMBL4112201 0.79 KDM4E (0.54) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL4118526 0.79 MAPT (0.66) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL4122854 0.79 KMT2A (0.56) KDM4ENPC1MAPTRAB9AKMT2A
SCHEMBL4106008 0.79 NPC1 (0.65) NPC1MAPTRAB9APKMKMT2A
SCHEMBL4113500 0.78 EPHX2 (0.58) KDM4EMAPTRAB9AKMT2AMEN1
SCHEMBL4112050 0.77 RAB9A (0.56) NPC1MAPTRAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804785-A2 DIARYL UREAS AS CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2007-07-11 EP claimed
WO-2006049941-A2 DIARYL UREAS AS CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2006-05-11 WO claimed