SCHEMBL5200951

SCHEMBL5200951

O=C(O)N[C@H](Cc1ccccc1F)CS(=O)(=O)Cl

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
KMT2A Q03164 6/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 3/20 0.40
LMNA P02545 2/20 0.40
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
KEAP1 Q14145 1/20 0.37
AKR1C3 P42330 1/20 0.36
CXCL8 P10145 1/20 0.35
GAA P10253 1/20 0.35
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5559459 0.83 CTRB1 (0.51) KMT2AALDH1A1CTSSCTSK
SCHEMBL4923623 0.81 CTSS (0.54) LMNACTSSCTSK
SCHEMBL14034476 0.80 MME (0.48) PPARGPPARAKMT2AALDH1A1MEN1
SCHEMBL6407838 0.75 CNR2 (0.45) KMT2AALDH1A1MEN1
SCHEMBL6407833 0.75 CNR2 (0.45) KMT2AALDH1A1MEN1
SCHEMBL5562553 0.71 CTRB1 (0.52) KMT2AALDH1A1CTSSCTSK
SCHEMBL4917131 0.69 CTSS (0.55) CTSSCTSK
SCHEMBL4917142 0.69 CTSS (0.55) CTSSCTSK
SCHEMBL5177986 0.69 NOTUM (0.47) KMT2AALDH1A1MEN1LMNAGAA
SCHEMBL28807054 0.68 PPARG (0.51) PPARGPPARAKMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858846-A1 DPP-IV INHIBITORS Santhera Pharmaceuticals (Schweiz) GmbH (CH) 2007-11-28 EP disclosed
WO-2006097175-A1 DPP-IV INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) AG (CH) 2006-09-21 WO disclosed