SCHEMBL5201006

SCHEMBL5201006

CS(=O)(=O)Nc1cc(OCC2=NCCN2)ccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 10/20 0.62
NISCH Q9Y2I1 5/20 0.51
DRD2 P14416 2/20 0.48
DRD3 P35462 2/20 0.48
ADRA1D P25100 8/20 0.47
ADRA1B P35368 8/20 0.47
ADRA2A P08913 7/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
DRD4 P21917 1/20 0.45
ADRA2C P18825 7/20 0.44
ADRA2B P18089 1/20 0.41
SCN9A Q15858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5204266 0.99 ADRA1A (0.61) ADRA1ANISCHDRD2DRD3ADRA1D
SCHEMBL5206394 0.87 ADRA1A (0.54) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5201523 0.86 NISCH (0.51) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5200760 0.86 NISCH (0.51) ADRA1ANISCHDRD2ADRA1DADRA1B
Hydrochloric Acid SCHEMBL5201136 0.86 ADRA1A (0.53) ADRA1ANISCHADRA1DADRA1BADRA2A
Hydrochloric Acid SCHEMBL5206302 0.85 ADRA1A (0.50) ADRA1ANISCHADRA1DADRA1BADRA2A
Hydrochloric Acid SCHEMBL5201887 0.85 ADRA1A (0.50) ADRA1ANISCHDRD2ADRA1DADRA1B
SCHEMBL14340664 0.83 ADRA1A (0.53) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5203763 0.81 ADRA1A (0.53) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5204186 0.81 ADRA1A (0.67) ADRA1ANISCHADRA1DADRA1BADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed