SCHEMBL5201127

SCHEMBL5201127

COC(=O)CNS(=O)(=O)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
MMP1 P03956 1/20 0.57
MMP2 P08253 1/20 0.57
MMP9 P14780 1/20 0.57
MMP8 P22894 1/20 0.57
MMP13 P45452 1/20 0.57
THRB P10828 1/20 0.57
ALDH1A1 P00352 3/20 0.56
CYP19A1 P11511 1/20 0.56
LMNA P02545 2/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
PKM P14618 1/20 0.52
SLC10A6 Q3KNW5 1/20 0.52
F2 P00734 2/20 0.51
PRSS1 P07477 2/20 0.51
PRSS2 P07478 2/20 0.51
PRSS3 P35030 2/20 0.51
TDP1 Q9NUW8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31120657 1.00 CA1 (0.57) CA1CA2MMP1MMP2MMP9
SCHEMBL18127253 0.88 CA1 (0.54) CA1CA2MMP1MMP2MMP9
SCHEMBL4644817 0.88 ALDH1A1 (0.56) CA1CA2MMP1MMP2MMP9
SCHEMBL4172892 0.86 KMT2A (0.56) CA1CA2MMP1MMP2MMP9
SCHEMBL18114379 0.84 MMP1 (0.62) CA1CA2MMP1MMP2MMP9
SCHEMBL7827745 0.84 MMP1 (0.62) CA1CA2MMP1MMP2MMP9
SCHEMBL15621323 0.84 CA1 (0.62) CA1CA2MMP1MMP2MMP9
SCHEMBL29096884 0.83 CYP19A1 (0.56) CA1CA2MMP1MMP2MMP9
SCHEMBL5693264 0.83 CA1 (0.51) CA1CA2MMP1MMP2MMP9
SCHEMBL18114431 0.83 CA1 (0.60) CA1CA2MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1400521-B1 PIPERAZINE COMPOUNDS KOWA CO (JP) 2007-11-07 EP disclosed
EP-1400521-A1 PIPERAZINE COMPOUNDS Kowa Co., Ltd. (JP) 2004-03-24 EP disclosed
US-6432957-B1 ANTIASTHMA; ANTIALLERGENS; RHEUMATIC DISEASES; ANTIINFLAMMATORY AGENTS KOWA CO., LTD. (JP) 2002-08-13 US disclosed