SCHEMBL5201186

SCHEMBL5201186

CS(=O)(=O)c1ccc(-n2nc(C(F)(F)F)nc2-c2ccc(OC(F)(F)F)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.53
PTGS1 P23219 6/20 0.52
CYP2C9 P11712 1/20 0.49
NPY5R Q15761 1/20 0.46
EPHX2 P34913 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6887276 0.90 PTGS2 (0.59) PTGS2PTGS1CYP2C9
SCHEMBL6885294 0.89 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL5202675 0.89 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL5205701 0.88 PTGS2 (0.51) PTGS2PTGS1CYP2C9
SCHEMBL5865485 0.87 PTGS2 (0.64) PTGS2PTGS1CYP2C9
SCHEMBL6885807 0.86 PTGS2 (0.61) PTGS2PTGS1CYP2C9
SCHEMBL5203782 0.86 PTGS2 (0.61) PTGS2PTGS1CYP2C9
SCHEMBL5205021 0.85 PTGS2 (0.57) PTGS2PTGS1CYP2C9
SCHEMBL5203055 0.85 PTGS2 (0.62) PTGS2PTGS1CYP2C9
SCHEMBL6884047 0.85 PTGS2 (0.62) PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539718-A4 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME CJ CORP (KR) 2007-08-01 EP claimed
US-7019144-B2 1,2,4-Triazole derivative, method for preparing the same, and pharmaceutical composition containing the same CJ CORP. (KR) 2006-03-28 US claimed
EP-1539718-A1 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME CJ Corporation (KR) 2005-06-15 EP claimed
WO-2004014878-A1 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME CJ CORPORATION (KR) 2004-02-19 WO claimed
EP-1539718-A4 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME CJ CORP (KR) 2007-08-01 EP disclosed
EP-1539718-A1 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME CJ Corporation (KR) 2005-06-15 EP disclosed
WO-2004014878-A1 1,2,4-TRIAZOLE DERIVATIVE, METHOD FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME CJ CORPORATION (KR) 2004-02-19 WO disclosed