SCHEMBL6885807

SCHEMBL6885807

CCOc1ccc(-n2nc(C(F)(F)F)nc2-c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.61
PTGS1 P23219 6/20 0.54
CYP2C9 P11712 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203782 1.00 PTGS2 (0.61) PTGS2PTGS1CYP2C9CA1CA2
SCHEMBL5202692 0.90 PTGS2 (0.67) PTGS2PTGS1CYP2C9CA1CA2
SCHEMBL6887276 0.88 PTGS2 (0.59) PTGS2PTGS1CYP2C9
SCHEMBL5202675 0.87 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL6885294 0.87 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL5201186 0.86 PTGS2 (0.53) PTGS2PTGS1CYP2C9
SCHEMBL5205203 0.86 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL14857230 0.86 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL5865485 0.85 PTGS2 (0.64) PTGS2PTGS1CYP2C9CA1CA2
SCHEMBL1115042 0.84 PTGS2 (0.47) PTGS2PTGS1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6803380-B1 NON-STEROIDAL ANTIINFLAMMATORY DRUGS LABORATOIRE THERAMEX (MC) 2004-10-12 US disclosed
EP-1246809-B1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM THERAMEX (MC) 2003-07-16 EP disclosed
EP-1246809-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2002-10-09 EP disclosed
WO-2001034577-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2001-05-17 WO disclosed
EP-1099695-A1 5-aryl-1H-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical compositions containing them LABORATOIRE THERAMEX S.A. (MC) 2001-05-16 EP disclosed