SCHEMBL5201360

SCHEMBL5201360

CC(C)(C)OC(=O)N1CCC(OC(=O)N2CCC(=O)C2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.46
PRMT5 O14744 2/20 0.44
WDR77 Q9BQA1 2/20 0.44
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
THRB P10828 1/20 0.43
HPGD P15428 1/20 0.43
PIK3CD O00329 1/20 0.43
GPR119 Q8TDV5 5/20 0.41
ESR2 Q92731 1/20 0.41
RECQL P46063 1/20 0.41
EPHX1 P07099 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
USP30 Q70CQ3 1/20 0.41
PTPN2 P17706 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6626522 0.88 MAPT (0.48) HPGDSMAPTKDM4ETHRBHPGD
SCHEMBL123032 0.83 ESR2 (0.54) MAPTKDM4ETHRBHPGDESR2
Methyl Alcohol SCHEMBL28603193 0.82 ESR2 (0.52) MAPTKDM4ETHRBHPGDESR2
SCHEMBL29703403 0.81 HPGD (0.64) MAPTKDM4ETHRBHPGDPIK3CD
SCHEMBL29703410 0.81 HPGD (0.64) MAPTKDM4ETHRBHPGDPIK3CD
SCHEMBL2721275 0.81 HPGD (0.64) MAPTKDM4ETHRBHPGDPIK3CD
SCHEMBL5201368 0.79 GPR119 (0.41) MAPTKDM4ETHRBHPGDGPR119
SCHEMBL6988508 0.78 HPGD (0.51) MAPTKDM4ETHRBHPGDPIK3CD
SCHEMBL13219346 0.78 HPGD (0.51) MAPTKDM4ETHRBHPGDPIK3CD
SCHEMBL65675 0.78 HPGD (0.51) MAPTKDM4ETHRBHPGDPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838687-A1 NON-ANILINIC DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS AstraZeneca AB (SE) 2007-10-03 EP disclosed
WO-2006073366-A1 NON-ANILINIC DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2006-07-13 WO disclosed