SCHEMBL5201781

SCHEMBL5201781

Cc1cc(C)c(OCC2=NCCN2)cc1NS(C)(=O)=O

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 11/20 0.58
NISCH Q9Y2I1 9/20 0.51
ADRA1D P25100 4/20 0.43
ADRA1B P35368 4/20 0.43
ADRA2A P08913 3/20 0.42
ADRA2C P18825 3/20 0.42
HTR1A P08908 2/20 0.42
ADRA2B P18089 2/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5204106 0.99 ADRA1A (0.57) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5202963 0.82 ADRA1A (0.60) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5206394 0.82 ADRA1A (0.54) ADRA1ANISCHADRA1DADRA1BADRA2A
Hydrochloric Acid SCHEMBL5201136 0.81 ADRA1A (0.53) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5201551 0.81 ADRA1A (0.64) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5202260 0.80 ADRA1A (0.66) ADRA1ANISCHADRA1DADRA1BADRA2A
Hydrochloric Acid SCHEMBL5203301 0.80 ADRA1A (0.62) ADRA1ANISCHADRA1DADRA1BADRA2A
Hydrochloric Acid SCHEMBL5201322 0.79 ADRA1A (0.65) ADRA1ANISCHADRA1DADRA1BADRA2A
SCHEMBL5201030 0.78 ADRA1A (0.80) ADRA1ANISCHADRA1DADRA1BADRA2A
Hydrochloric Acid SCHEMBL5200769 0.76 ADRA1A (0.55) ADRA1ANISCHADRA1DADRA1BADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed