SCHEMBL5201851

SCHEMBL5201851

[CH2]CCC(=O)N(Cc1ccccc1F)Nc1ccc(Cl)cc1Oc1cccc(CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
NPSR1 Q6W5P4 3/20 0.39
HTT P42858 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 2/20 0.36
P2RX4 Q99571 1/20 0.36
MAPT P10636 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GAA P10253 1/20 0.35
PPARG P37231 2/20 0.35
PPARD Q03181 2/20 0.35
PPARA Q07869 2/20 0.35
GLS O94925 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
EPAS1 Q99814 1/20 0.33
ANO1 Q5XXA6 1/20 0.33
TP53 P04637 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833900 0.79 ALDH1A1 (0.43) ALDH1A1NPSR1HTTLMNAPOLB
SCHEMBL5208884 0.79 KDM4E (0.41) ALDH1A1NPSR1HTTLMNAPOLB
SCHEMBL5203560 0.79 ALDH1A1 (0.45) ALDH1A1NPSR1HTTLMNAPOLB
SCHEMBL5204994 0.75 ALDH1A1 (0.40) ALDH1A1NPSR1HTTLMNAPOLB
SCHEMBL5203418 0.74 ALDH1A1 (0.40) ALDH1A1NPSR1HTTLMNAPOLB
SCHEMBL5205300 0.73 PPARG (0.41) ALDH1A1HTTKDM4ESMN1; SMN2GAA
SCHEMBL5205860 0.72 PPARG (0.42) HTTSMN1; SMN2GAAPPARGPPARD
SCHEMBL5202191 0.72 PPARG (0.42) ALDH1A1HTTSMN1; SMN2PPARGPPARD
SCHEMBL5205234 0.72 TSHR (0.46) SMN1; SMN2GAAPPARGPPARDPPARA
SCHEMBL5205312 0.71 PPARG (0.40) ALDH1A1HTTKDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed