SCHEMBL5202777

SCHEMBL5202777

N#Cc1ccc2c(N3CCN(CCCCc4c[nH]c5ccc(C(=O)O)cc45)CC3)cc(=O)oc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.56
DRD2 P14416 3/20 0.56
ADRA2A P08913 2/20 0.56
ADRA2C P18825 2/20 0.56
SLC6A2 P23975 2/20 0.56
ADRA1D P25100 2/20 0.56
SLC6A4 P31645 2/20 0.56
HTR7 P34969 2/20 0.56
ADRA1A P35348 2/20 0.56
ADRA1B P35368 2/20 0.56
SLC6A3 Q01959 2/20 0.56
ADRA2B P18089 1/20 0.56
KCNH2 Q12809 1/20 0.56
ADRB2 P07550 1/20 0.55
DRD4 P21917 1/20 0.55
FPR3 P25089 1/20 0.55
HTR1D P28221 1/20 0.55
HTR1B P28222 1/20 0.55
GPR183 P32249 1/20 0.55
HRH1 P35367 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7787585 0.95 HTR1A (0.51) HTR1ADRD2ADRA2AADRA2CSLC6A2
SCHEMBL7788884 0.91 HTR1A (0.54) HTR1ADRD2ADRA2AADRA2CSLC6A2
SCHEMBL5203156 0.88 HTR1A (0.54) HTR1ASLC6A4HTR7ADRA1AKCNH2
SCHEMBL5204246 0.88 KDM4E (0.51) HTR1AADRA2AADRA2CADRA1DADRA1A
SCHEMBL5203306 0.88 HTR1A (0.50) HTR1AADRA2AADRA2CADRA1DSLC6A4
SCHEMBL5203078 0.87 KDM4E (0.56) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL5204281 0.86 ADRA2A (0.60) HTR1ADRD2ADRA2AADRA2CADRA1D
SCHEMBL8140840 0.86 HTR1A (0.54) HTR1ADRD2ADRA2AADRA2CSLC6A2
SCHEMBL7784868 0.86 HTR1A (0.49) HTR1ADRD2ADRA2AADRA2CSLC6A2
SCHEMBL5201581 0.86 HTR1A (0.63) HTR1ADRD2KCNH2HTR6HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998474-B1 PIPERAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-07 EP disclosed
US-6251908-B1 Piperazine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2001-06-26 US disclosed