SCHEMBL5202957

SCHEMBL5202957

COc1ccc(C(=O)Nc2cccc(C(=O)Cl)c2)cc1OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.80
POLB P06746 4/20 0.71
MEN1 O00255 5/20 0.65
KMT2A Q03164 5/20 0.65
RAB9A P51151 5/20 0.65
NPC1 O15118 4/20 0.65
SMN1; SMN2 Q16637 3/20 0.65
LMNA P02545 2/20 0.65
MAPT P10636 2/20 0.65
L3MBTL1 Q9Y468 1/20 0.62
NQO2 P16083 1/20 0.62
CASP3 P42574 1/20 0.62
SENP7 Q9BQF6 1/20 0.62
TP53 P04637 2/20 0.60
PKM P14618 1/20 0.59
MAPK14 Q16539 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
SETD7 Q8WTS6 1/20 0.57
PDE4D Q08499 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203706 0.83 KCNK9 (0.76) ALDH1A1MEN1KMT2ARAB9ANPC1
SCHEMBL4248720 0.83 RXFP1 (0.76) ALDH1A1POLBMEN1KMT2ARAB9A
SCHEMBL14363225 0.83 POLB (0.75) ALDH1A1POLBMEN1KMT2ARAB9A
SCHEMBL4141962 0.83 MEN1 (0.89) ALDH1A1POLBMEN1KMT2ARAB9A
SCHEMBL31331620 0.82 ALDH1A1 (0.73) ALDH1A1POLBMEN1KMT2ARAB9A
Hydrochloric Acid SCHEMBL9638131 0.81 MEN1 (0.86) ALDH1A1POLBMEN1KMT2ARAB9A
SCHEMBL29521706 0.81 TSHR (0.70) ALDH1A1POLBSMN1; SMN2LMNAMAPT
SCHEMBL184025 0.81 TSHR (0.70) ALDH1A1POLBSMN1; SMN2LMNAMAPT
SCHEMBL4098536 0.80 CHEK1 (0.84) ALDH1A1POLBMEN1KMT2ARAB9A
SCHEMBL13561150 0.79 MAPT (0.68) ALDH1A1POLBMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087946-B1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2007-01-10 EP disclosed
CN-1168720-C Aryl alkanoylpyridazines Ĭ��ר���ɷ����޹�˾ 2004-09-29 CN disclosed
US-6417188-B1 ENZYME INHIBITORS OF PHOSPHODIESTERASE MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-07-09 US disclosed
CN-1305465-A Aryl alkanoylpyridazines MERCK PATENT GMBH (DE) 2001-07-25 CN disclosed
EP-1087946-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2001-04-04 EP disclosed
WO-1999065880-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 1999-12-23 WO disclosed