SCHEMBL5203427

SCHEMBL5203427

CS(=O)(=O)Nc1cc(CC2=NCCN2)ccc1F

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.48
TAAR1 Q96RJ0 3/20 0.47
CYP2D6 P10635 2/20 0.47
NFKB1 P19838 1/20 0.47
ADRA1D P25100 9/20 0.46
ADRA1A P35348 9/20 0.46
ADRA1B P35368 9/20 0.46
ADRA2C P18825 8/20 0.46
ADRA2A P08913 7/20 0.46
HTR1D P28221 5/20 0.46
HTR1B P28222 4/20 0.45
ADRA2B P18089 2/20 0.45
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5200588 0.99 RAD52 (0.47) RAD52TAAR1CYP2D6NFKB1ADRA1D
SCHEMBL4992620 0.90 ADRA1D (0.49) RAD52TAAR1CYP2D6NFKB1ADRA1D
SCHEMBL5200888 0.86 RAD52 (0.49) RAD52TAAR1CYP2D6NFKB1ADRA1D
SCHEMBL5203274 0.85 ADRA1A (0.55) RAD52TAAR1CYP2D6NFKB1ADRA1D
SCHEMBL5203954 0.85 ADRA1A (0.51) RAD52TAAR1CYP2D6NFKB1ADRA1D
Hydrochloric Acid SCHEMBL5201249 0.85 RAD52 (0.48) RAD52TAAR1CYP2D6NFKB1ADRA1D
Bromide SCHEMBL5200819 0.84 ADRA1A (0.56) RAD52TAAR1CYP2D6NFKB1ADRA1D
Hydrochloric Acid SCHEMBL5205831 0.84 ADRA1A (0.50) RAD52TAAR1CYP2D6NFKB1ADRA1D
SCHEMBL4993472 0.84 RAD52 (0.49) RAD52TAAR1CYP2D6NFKB1ADRA1D
SCHEMBL5200788 0.83 HTR1B (0.51) RAD52TAAR1CYP2D6NFKB1ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed