SCHEMBL5204517

SCHEMBL5204517

O=C(Nc1cccc(CN2CCCCC2)c1)C1=Cc2cc(-c3ccccc3)ccc2CC1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 16/20 0.58
MCHR1 Q99705 1/20 0.53
FAAH O00519 1/20 0.51
CDK5 Q00535 1/20 0.49
CDK5R1 Q15078 1/20 0.49
SLC2A1 P11166 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674643 0.90 CCR5 (0.68) CCR5MCHR1
SCHEMBL5208758 0.90 CCR5 (0.68) CCR5MCHR1
SCHEMBL5211618 0.89 CCR5 (0.69) CCR5MCHR1
SCHEMBL7674608 0.83 CCR5 (0.69) CCR5
SCHEMBL5205976 0.83 CCR5 (0.58) CCR5MCHR1
SCHEMBL5209488 0.82 CCR5 (0.69) CCR5MCHR1
SCHEMBL5203702 0.81 CCR5 (0.69) CCR5
Iodide SCHEMBL7682596 0.81 CCR5 (0.83) CCR5
SCHEMBL5208454 0.77 CCR5 (0.70) CCR5MCHR1
SCHEMBL5207505 0.77 CCR5 (0.74) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed