SCHEMBL5205380

SCHEMBL5205380

Nc1nc(-c2ccccn2)c2c(-c3ccccn3)cccc2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
ALOX15 P16050 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
TGFBR1 P36897 4/20 0.44
ADORA2A P29274 7/20 0.43
LMNA P02545 2/20 0.42
CCR1 P32246 2/20 0.42
CCR5 P51681 2/20 0.42
CCR8 P51685 2/20 0.42
ADORA1 P30542 1/20 0.42
TP53 P04637 1/20 0.42
ALPL P05186 1/20 0.42
HSP90AA1 P07900 1/20 0.42
ALPI P09923 1/20 0.42
ALPG P10696 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25430300 0.84 KDM4E (0.51) KDM4EALOX15L3MBTL1TGFBR1ADORA2A
SCHEMBL367849 0.78 ADORA2A (0.61) KDM4EALOX15L3MBTL1TGFBR1ADORA2A
SCHEMBL30455036 0.75 KCNH2 (0.43) KDM4EALOX15L3MBTL1TGFBR1LMNA
SCHEMBL26260016 0.73 KDM4E (0.58) KDM4EALOX15L3MBTL1TGFBR1LMNA
SCHEMBL6824538 0.72 KDM4E (0.50) KDM4EALOX15L3MBTL1TGFBR1ADORA2A
Dipyridyl SCHEMBL29167113 0.70 KDM4E (0.79) KDM4EALOX15L3MBTL1LMNACCR1
SCHEMBL13728155 0.70 NPC1 (0.52) KDM4EALOX15L3MBTL1TGFBR1LMNA
SCHEMBL13726458 0.69 TGFBR1 (0.49) KDM4EALOX15L3MBTL1TGFBR1LMNA
SCHEMBL4106450 0.69 ADORA2A (0.47) KDM4EALOX15L3MBTL1TGFBR1ADORA2A
SCHEMBL2061612 0.68 KDM4E (0.70) KDM4EALOX15L3MBTL1TGFBR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742634-A1 POLYCYCLIC PYRIMIDINES AS POTASSIUM ION CHANNEL MODULATORS ICAgen, Incorporated (US) 2007-01-17 EP disclosed
WO-2005099711-A1 POLYCYCLIC PYRIMIDINES AS POTASSIUM ION CHANNEL MODULATORS ICAGEN, INC. (US) 2005-10-27 WO disclosed