Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL5205518

COc1cc(CN(C(=O)CCC(=O)NC2CCc3ccccc32)c2ccccc2Oc2cccc(CN)c2)cc(OC)c1OC.O=C(O)C(F)(F)F

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.43
HCRTR2 O43614 3/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
CCR8 P51685 1/20 0.37
ADORA2A P29274 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
TSPO P30536 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5206411 0.93 HCRTR1 (0.39) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5202626 0.91 ALDH1A1 (0.42) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5205258 0.90 TAOK1 (0.39) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5202194 0.90 HCRTR1 (0.43) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5202074 0.89 TAOK1 (0.39) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5206105 0.89 CFD (0.38) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5208207 0.88 HCRTR1 (0.37) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5206323 0.87 HCRTR1 (0.36) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5202445 0.87 DHODH (0.39) HCRTR1HCRTR2MEN1KMT2ASMN1; SMN2
Trifluoroacetic Acid SCHEMBL5205747 0.87 PARP1 (0.37) HCRTR1HCRTR2MEN1KMT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed