SCHEMBL5205767

SCHEMBL5205767

CCOc1ccc(C2=NN(C(=O)c3ccc(N)cc3)CCC2)cc1OCC

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PGR P06401 14/20 0.52
ALDH1A1 P00352 4/20 0.50
GAA P10253 1/20 0.50
POLB P06746 1/20 0.49
LMNA P02545 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PKM P14618 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MAOB P27338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3920897 0.95 ALDH1A1 (0.52) PGRALDH1A1GAAPOLBLMNA
SCHEMBL3921282 0.89 ALDH1A1 (0.52) PGRALDH1A1GAAPOLBLMNA
SCHEMBL6584572 0.88 NPC1 (0.45) PGRALDH1A1GAAPOLBMAPT
SCHEMBL3927077 0.87 ALDH1A1 (0.50) PGRALDH1A1GAAPOLBLMNA
SCHEMBL6604789 0.86 MAOB (0.59) PGRALDH1A1GAAPOLBLMNA
SCHEMBL13210796 0.86 ALDH1A1 (0.53) PGRALDH1A1GAAPOLBLMNA
SCHEMBL5202716 0.84 ALDH1A1 (0.49) PGRALDH1A1GAAPOLBLMNA
SCHEMBL143747 0.84 ALDH1A1 (0.48) PGRALDH1A1GAAPOLBLMNA
SCHEMBL6581799 0.83 NPC1 (0.45) PGRALDH1A1POLBLMNAMAPT
SCHEMBL13210770 0.83 ALDH1A1 (0.52) PGRALDH1A1GAAPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087946-B1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2007-01-10 EP disclosed
CN-1168720-C Aryl alkanoylpyridazines Ĭ��ר���ɷ����޹�˾ 2004-09-29 CN disclosed
US-6417188-B1 ENZYME INHIBITORS OF PHOSPHODIESTERASE MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-07-09 US disclosed
CN-1305465-A Aryl alkanoylpyridazines MERCK PATENT GMBH (DE) 2001-07-25 CN disclosed
EP-1087946-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2001-04-04 EP disclosed
WO-1999065880-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 1999-12-23 WO disclosed