SCHEMBL6584572

SCHEMBL6584572

CCOc1cc(C2=NN(C(=O)c3ccc(NC(=O)c4ccc(N)cc4)cc3)CCC2)ccc1OC

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
TP53 P04637 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
POLB P06746 3/20 0.45
ALDH1A1 P00352 2/20 0.45
ABCB1 P08183 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
MAOB P27338 1/20 0.43
PGR P06401 3/20 0.42
MAPT P10636 3/20 0.42
GAA P10253 2/20 0.42
CASP1 P29466 1/20 0.42
KMT2A Q03164 3/20 0.42
CFTR P13569 2/20 0.42
MEN1 O00255 2/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581784 0.92 ALDH1A1 (0.55) NPC1RAB9ATP53SMN1; SMN2POLB
SCHEMBL6582201 0.92 GAA (0.51) NPC1RAB9ATP53SMN1; SMN2POLB
SCHEMBL6587589 0.92 ALDH1A1 (0.52) TP53SMN1; SMN2POLBALDH1A1MAOB
SCHEMBL3920897 0.92 ALDH1A1 (0.52) SMN1; SMN2POLBALDH1A1MAOBPGR
SCHEMBL6581232 0.92 POLB (0.44) NPC1RAB9ATP53SMN1; SMN2POLB
SCHEMBL6581799 0.92 NPC1 (0.45) NPC1RAB9ATP53SMN1; SMN2POLB
SCHEMBL6601230 0.92 HTT (0.47) SMN1; SMN2POLBALDH1A1MAOBMAPT
SCHEMBL6581226 0.92 PGR (0.54) SMN1; SMN2POLBALDH1A1MAOBPGR
Hydrochloric Acid SCHEMBL7646217 0.91 HTT (0.47) SMN1; SMN2POLBALDH1A1MAOBMAPT
SCHEMBL143747 0.91 ALDH1A1 (0.48) SMN1; SMN2POLBALDH1A1MAOBPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed
EP-1194411-A1 BENZOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001004099-A1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2001-01-18 WO disclosed