SCHEMBL5206017

SCHEMBL5206017

O=C(O)C1=Cc2cc(-c3ccc4c(c3)OCO4)ccc2SCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
MAPK1 P28482 1/20 0.41
EDNRB P24530 2/20 0.40
EDNRA P25101 2/20 0.40
NPC1 O15118 6/20 0.40
RAB9A P51151 5/20 0.40
PTGER4 P35408 1/20 0.39
KMT2A Q03164 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
SLC13A5 Q86YT5 1/20 0.39
CTNNB1 P35222 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
SRD5A2 P31213 1/20 0.38
TP53 P04637 1/20 0.38
DHODH Q02127 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5206762 0.86 NPC1 (0.43) ALDH1A1MAPK1NPC1RAB9AKMT2A
SCHEMBL5204016 0.80 ALDH1A1 (0.45) ALDH1A1MAPK1NPC1RAB9AKMT2A
SCHEMBL3499129 0.80 MCL1 (0.40) ALDH1A1KMT2AHPGDMAPTDHODH
SCHEMBL7682561 0.77 ALDH1A1 (0.42) ALDH1A1KDM4EHPGDMAPTDHODH
SCHEMBL5206801 0.75 AOC3 (0.42) ALDH1A1NPC1RAB9AKMT2AKDM4E
SCHEMBL7975031 0.75 ALDH1A1 (0.40) ALDH1A1MAPK1EDNRBEDNRANPC1
SCHEMBL7250245 0.70 HPGD (0.38) ALDH1A1KDM4EHPGDMAPT
SCHEMBL2945422 0.68 ALDH1A1 (0.73) ALDH1A1MAPK1NPC1RAB9APTGER4
SCHEMBL3498192 0.66 MCL1 (0.42) ALDH1A1MAPK1LMNAMAPTDHODH
SCHEMBL7683946 0.66 KDM4E (0.43) NPC1RAB9AKDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed