SCHEMBL7250245

SCHEMBL7250245

O=C(O)C1=Cc2ccccc2SCC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.38
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RYR2 Q92736 3/20 0.36
ALOX5 P09917 2/20 0.36
GSK3B P49841 1/20 0.36
NOTUM Q6P988 2/20 0.35
MCL1 Q07820 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
TBXAS1 P24557 1/20 0.33
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8651466 0.85 ALOX5 (0.38) HPGDMAPTALDH1A1PLA2G1BATG4B
SCHEMBL214797 0.82 NOTUM (0.40) HPGDMAPTALDH1A1RYR2ALOX5
SCHEMBL7251900 0.81 CA12 (0.46) HPGDMAPTALDH1A1PLA2G1BATG4B
SCHEMBL7247717 0.77 TSHR (0.42) HPGDMAPTALDH1A1PLA2G1BATG4B
SCHEMBL7382853 0.72 MAPT (0.31) HPGDMAPTALDH1A1PLA2G1BATG4B
SCHEMBL29427899 0.71 MAOA (0.49) HPGDALDH1A1ALOX5NOTUMKDM4E
SCHEMBL983738 0.71 MAOA (0.49) HPGDALDH1A1ALOX5NOTUMKDM4E
SCHEMBL7682561 0.70 ALDH1A1 (0.42) HPGDMAPTALDH1A1RYR2ALOX5
SCHEMBL10334576 0.70 KDM4E (0.48) ALDH1A1KDM4E
SCHEMBL5206017 0.70 ALDH1A1 (0.41) HPGDMAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566535-B1 Causing an orthohalogenobenzaldehyde or derivative to react with a propanethiol having an electron-attracting group at its 4- position. TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-20 US disclosed
EP-1184381-A1 PROCESSES FOR THE PREPARATION OF 2,3-DIHYDROTHIEPINE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2002-03-06 EP disclosed
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed