SCHEMBL5207901

SCHEMBL5207901

CN1CCC(CN2CCN(C(=O)CCc3oc(Cc4ccccc4)nc3-c3ccc(Cl)cc3)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 1/20 0.46
CACNA1B Q00975 1/20 0.46
CACNB1 Q02641 1/20 0.46
CACNA1C Q13936 1/20 0.46
TACR1 P25103 6/20 0.46
POLB P06746 1/20 0.45
HTT P42858 3/20 0.42
HRH3 Q9Y5N1 1/20 0.42
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TACR2 P21452 1/20 0.39
HTR7 P34969 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CACNA1G O43497 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5212688 0.88 TACR1 (0.50) CACNA2D1CACNA1BCACNB1CACNA1CTACR1
Hydrochloric Acid SCHEMBL5209960 0.88 TACR1 (0.49) CACNA2D1CACNA1BCACNB1CACNA1CTACR1
SCHEMBL5210242 0.84 TACR1 (0.47) CACNA2D1CACNA1BCACNB1CACNA1CTACR1
SCHEMBL5213964 0.84 KMT2A (0.44) TACR1POLBHTTMAPTTSHR
SCHEMBL5210692 0.83 CACNA2D1 (0.48) CACNA2D1CACNA1BCACNB1CACNA1CHTT
SCHEMBL5212036 0.83 TACR1 (0.46) CACNA2D1CACNA1BCACNB1CACNA1CTACR1
SCHEMBL5210396 0.82 MEN1 (0.43) TACR1POLBHTTMAPTALDH1A1
SCHEMBL5213743 0.82 TACR1 (0.49) CACNA2D1CACNA1BCACNB1CACNA1CTACR1
SCHEMBL5212616 0.82 TACR1 (0.45) CACNA2D1CACNA1BCACNB1CACNA1CTACR1
SCHEMBL5207975 0.81 TACR1 (0.45) CACNA2D1CACNA1BCACNB1CACNA1CTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7183276-B2 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US disclosed
US-20050090534-A1 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-04-28 US disclosed
EP-1486490-A1 AZOLE COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2004-12-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050090534-A1 Azole compounds AHR, NR0B2, NR2C2 CACNA2D1 4406/4885CACNA1B 1842/4885CACNB1 3052/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.