SCHEMBL5208873

SCHEMBL5208873

C[SiH](C)C(C)(C)COCc1ccc(N)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.37
ALDH1A1 P00352 4/20 0.37
APP P05067 1/20 0.36
GFER P55789 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.34
MAPT P10636 3/20 0.34
RAB9A P51151 3/20 0.34
GAA P10253 1/20 0.34
MAOA P21397 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TACR1 P25103 1/20 0.33
CYP19A1 P11511 2/20 0.33
NPC1 O15118 2/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6421635 0.82 APP (0.44) ALDH1A1APPCYP3A4IDO1
SCHEMBL481256 0.82 IDO1 (0.42) MAOBALDH1A1APPKDM4EMAPT
SCHEMBL28552350 0.78 ALDH1A1 (0.35) ALDH1A1
SCHEMBL8710528 0.78 ALDH1A1 (0.37) MAOBALDH1A1TDP1MAPTRAB9A
SCHEMBL18795029 0.76 HDAC3 (0.36) ALDH1A1
SCHEMBL234606 0.73 ALDH1A1 (0.55) MAOBALDH1A1APPGFERCYP3A4
SCHEMBL2561171 0.73 ALDH1A1 (0.58) MAOBALDH1A1APPGFERCYP3A4
SCHEMBL7337658 0.72 MAOB (0.35) MAOBALDH1A1APPGFERCYP3A4
SCHEMBL21493100 0.72 KMT2A (0.31) ALDH1A1RAB9ASMN1; SMN2
SCHEMBL5442094 0.71 CYP2A6 (0.34) MAOBALDH1A1KDM4EMAPTMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6376536-B1 VIRICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-04-23 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
EP-1104416-A2 QUATERNARY AMMONIUM SALTS AND THEIR USE AS ANTI-HIV AGENTS Takeda Chemical Industries, Ltd. (JP) 2001-06-06 EP disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
EP-1040103-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
EP-1039899-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
US-6096780-A ANTIVIRAL COMPOUND USEFUL FOR TREATING HIV VIRUSES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-08-01 US disclosed
WO-2000010965-A2 QUATERNARY AMMONIUM SALTS AND THEIR USE AS ANTI-HIV AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-03-02 WO disclosed
WO-1999032100-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed
WO-1999032468-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed