SCHEMBL5209233

SCHEMBL5209233

C#CC(O)c1c(-c2ccco2)nn2c(Cl)cccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.41
MEN1 O00255 6/20 0.41
MAPT P10636 5/20 0.41
BLM P54132 4/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 7/20 0.33
KDM4E B2RXH2 6/20 0.33
POLB P06746 4/20 0.33
RECQL P46063 4/20 0.33
L3MBTL1 Q9Y468 4/20 0.33
HPGD P15428 4/20 0.33
PTPN7 P35236 3/20 0.33
ALOX12 P18054 3/20 0.33
PKM P14618 3/20 0.33
TDP1 Q9NUW8 3/20 0.33
HSD17B10 Q99714 3/20 0.33
LMNA P02545 2/20 0.33
ALOX15 P16050 2/20 0.33
CASP1 P29466 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5212546 0.81 ALDH1A1 (0.32) KMT2AMEN1TSHRALDH1A1POLB
SCHEMBL5209264 0.81 MAPK14 (0.30) MAPK14
SCHEMBL5211466 0.76 KMT2A (0.38) KMT2AMEN1MAPTBLMTSHR
SCHEMBL6108701 0.75 CFTR (0.35) MAPTALDH1A1MAPK14NPC1NPSR1
SCHEMBL5943206 0.75 PIK3CD (0.34) MAPTTSHRKDM4EPOLBRECQL
SCHEMBL6105571 0.74 MAPK14 (0.37) KMT2AMEN1MAPTALDH1A1KDM4E
SCHEMBL5212439 0.74 MAPT (0.45) KMT2AMEN1MAPTBLMTSHR
SCHEMBL5208134 0.71 MEN1 (0.42) KMT2AMEN1MAPTBLMTSHR
SCHEMBL5449798 0.64 MAPK14 (0.51) RECQLADORA3ADORA2AADORA1MAPK14
SCHEMBL31352124 0.61 RECQL (0.38) RECQLTDP1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453830-B1 PYRAZOLO-PYRIDINE DERIVATIVES AS ANTIHERPES AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-12 EP disclosed
US-20070161653-A1 Pyrazolo-Pyridine Derivatives As Antiherpes Agents GUDMUNDSSON KRISTJAN 2007-07-12 US disclosed
US-7199120-B2 Pyrazolo-pyridine derivatives as antiherpes agents SMITHKLINE BEECHAM CORPORATION (US) 2007-04-03 US disclosed
US-20040248903-A1 Pyrazolo-pyridine derivatives as antiherpes agents SMITHKLINE BEECHAM CORPORATION 2004-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070161653-A1 Pyrazolo-Pyridine Derivatives As Antiherpes Agents HRH4, HRH2, HRH1 KMT2A 1758/4885MEN1 2749/4885MAPT 1616/4885
US-20040248903-A1 Pyrazolo-pyridine derivatives as antiherpes agents HRH4, HRH1, HRH2 KMT2A 1694/4885MEN1 2302/4885MAPT 1457/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.