SCHEMBL5209433

SCHEMBL5209433

CC1(C)OCc2cc([C@@H](O)CNCCc3ccc4c(c3)O[C@H](COCc3cccc(C(N)=O)c3)CO4)ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 13/20 0.38
ADRB1 P08588 12/20 0.38
ADRB2 P07550 11/20 0.38
ADRA1D P25100 5/20 0.38
ADRA1A P35348 5/20 0.38
ADRA1B P35368 5/20 0.38
ALDH1A1 P00352 2/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SLC22A1 O15245 1/20 0.33
CHRM2 P08172 1/20 0.33
CYP3A4 P08684 1/20 0.33
CHRM1 P11229 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
SLC6A4 P31645 1/20 0.33
OPRM1 P35372 1/20 0.33
SLC6A3 Q01959 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5209443 1.00 ADRB3 (0.38) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5209050 0.91 ADRB2 (0.42) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5209039 0.91 ADRB2 (0.42) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5212693 0.90 ADRB2 (0.39) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5209792 0.90 ADRB2 (0.39) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5212863 0.88 ADRB3 (0.35) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5212232 0.88 ADRB2 (0.35) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5212239 0.88 ADRB2 (0.35) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5943664 0.87 ADRB2 (0.39) ADRB3ADRB1ADRB2ADRA1DADRA1A
SCHEMBL5943639 0.86 ADRB2 (0.36) ADRB3ADRB1ADRB2ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554264-B1 MEDICINAL ARYLETHANOLAMINE COMPOUNDS GLAXO GROUP LTD (GB) 2007-08-08 EP disclosed