SCHEMBL5215845

SCHEMBL5215845

COCOC(CO)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.44
CYP19A1 P11511 2/20 0.38
TRPA1 O75762 1/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 1/20 0.37
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5220341 0.82 AOC3 (0.44) AOC3SLC6A2SLC6A4SLC6A3IDO1
SCHEMBL8171991 0.82 CYP19A1 (0.38) CYP19A1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL2065578 0.81 GSR (0.47) CYP19A1TRPA1SLC6A4HPGD
SCHEMBL2065580 0.81 GSR (0.47) CYP19A1TRPA1SLC6A4HPGD
SCHEMBL5350841 0.79 AOC3 (0.41) AOC3CYP19A1SLC6A2SLC6A4SLC6A3
SCHEMBL5350840 0.79 AOC3 (0.42) AOC3CYP19A1ALDH1A1MAPTHTT
SCHEMBL5350835 0.74 AOC3 (0.38) AOC3CYP19A1SLC6A2SLC6A4SLC6A3
SCHEMBL1154822 0.70 CYP3A4 (0.47)
SCHEMBL4729832 0.70 AOC3 (0.39) AOC3TRPA1SLC6A2SLC6A4ALDH1A1
SCHEMBL5223462 0.68 AOC3 (0.37) AOC3TRPA1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed