SCHEMBL5216772

SCHEMBL5216772

COc1ccc(-c2ccc(C34C=CCN(CC3)C4)cn2)cc1OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 7/20 0.38
TNF P01375 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
HSD17B10 Q99714 1/20 0.35
GAK O14976 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
KDM1A O60341 2/20 0.34
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL4481380 0.99 FYN (0.38) FYNTNFSMN1; SMN2KDM4EALDH1A1
SCHEMBL4463735 0.86 RXFP1 (0.39) FYNSMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL2678945 0.83 FYN (0.43) FYNTNFSMN1; SMN2KDM4EALDH1A1
SCHEMBL4475112 0.82 CHRNA7 (0.37) KDM1A
SCHEMBL4461401 0.81 ALOX5AP (0.31) KDM1A
SCHEMBL4465250 0.81 KDM1A (0.40) SMN1; SMN2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL4470449 0.80 SLC6A2 (0.38) FYNKDM4EALDH1A1KDM1ACYP2D6
SCHEMBL4463819 0.79 HSD11B1 (0.38)
SCHEMBL5223011 0.79 FYN (0.40) FYNTNFSMN1; SMN2KDM4EALDH1A1
SCHEMBL2678759 0.79 FYN (0.42) FYNTNFSMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465893-B1 DERIVATIVES OF 5-(PYRIDIN-3-YL)-1-AZABICYCLO (3.2.1) OCTANE, THE PREPARATION THEREOF AND THE APPLICATION OF SAME IN THERAPEUTICS SANOFI AVENTIS (FR) 2007-02-28 EP claimed