SCHEMBL5220629

SCHEMBL5220629

CCNc1cc(C(=O)O)c(F)c(N2CCCCS2(O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.43
BACE2 Q9Y5Z0 16/20 0.43
CTSD P07339 15/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.34
AVPR2 P30518 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223182 0.97 BACE1 (0.40) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5219939 0.89 BACE1 (0.43) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5220634 0.89 BACE1 (0.52) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5221778 0.85 BACE1 (0.41) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5223174 0.85 BACE1 (0.49) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5221190 0.85 CTSD (0.34) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5223783 0.83 CTSD (0.30) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5218910 0.83 MCL1 (0.34) BACE1BACE2CTSDCYP3A4CYP2D6
SCHEMBL5222895 0.79 MCL1 (0.35)
SCHEMBL5219943 0.78 BACE1 (0.53) BACE1BACE2CTSDCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed