SCHEMBL5221894

SCHEMBL5221894

CCn1ncc2c(N3CCCC3=O)cc(C(=O)OC)cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.49
CTSD P07339 3/20 0.49
BACE2 Q9Y5Z0 3/20 0.49
CYP2C9 P11712 3/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.36
PTGER3 P43115 2/20 0.36
HPGD P15428 3/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CREBBP Q92793 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5219279 0.90 CTSD (0.51) BACE1CTSDBACE2CYP2C9CYP3A4
SCHEMBL5216173 0.80 CTSD (0.49) BACE1CTSDBACE2CYP2C9CYP3A4
SCHEMBL5222810 0.79 BACE1 (0.51) BACE1CTSDBACE2CYP2C9CYP3A4
SCHEMBL5218380 0.79 PIK3C3 (0.39) BACE1CTSDBACE2MAPTPTGER3
SCHEMBL5218370 0.79 PTGER3 (0.37) BACE1CTSDBACE2MAPTPTGER3
SCHEMBL5221959 0.78 KDM4E (0.41) MAPTPTGER3HPGDALDH1A1KDM4E
SCHEMBL5218022 0.76 BACE1 (0.50) BACE1CTSDBACE2CYP2C9CYP3A4
SCHEMBL5379366 0.76 SCN9A (0.43) BACE1CTSDBACE2SIGMAR1
SCHEMBL15910578 0.75 KDM4E (0.48) CYP2C9MAPTPTGER3ALDH1A1KDM4E
SCHEMBL5222417 0.75 CYP2C9 (0.42) BACE1CTSDBACE2CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed