SCHEMBL5223147

SCHEMBL5223147

COc1cc2c(Oc3ccccc3F)ccnc2cc1OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MET P08581 12/20 0.58
KDR P35968 2/20 0.58
MST1R Q04912 2/20 0.58
SRC P12931 1/20 0.54
TGFBR1 P36897 1/20 0.54
HGF P14210 1/20 0.53
AXL P30530 2/20 0.53
FGFR2 P21802 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL2063874 0.99 MET (0.57) METKDRMST1RSRCTGFBR1
SCHEMBL13787641 0.89 MET (0.59) METKDRMST1RSRCTGFBR1
SCHEMBL13739661 0.89 SRC (0.60) METKDRMST1RSRCTGFBR1
SCHEMBL30216641 0.88 MET (0.58) METKDRMST1RHGFAXL
SCHEMBL31412927 0.88 AXL (0.61) METKDRMST1RHGFAXL
SCHEMBL372031 0.88 AXL (0.61) METKDRMST1RHGFAXL
SCHEMBL21408242 0.88 MET (0.58) METKDRMST1RHGFAXL
SCHEMBL6592222 0.88 KDM1A (0.56) FGFR2
SCHEMBL10296328 0.88 KDM1A (0.56) FGFR2
SCHEMBL16933077 0.87 AXL (0.60) METKDRMST1RHGFAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1827434-A2 QUINOLINES AND QUINAZOLINE ANALOGS AND THEIR USE AS MEDICAMENTS FOR TREATING CANCER Amgen Inc. (US) 2007-09-05 EP disclosed
WO-2006060318-A2 QUINOLINES AND QUINAZOLINE ANALOGS AND THEIR USE AS MEDICAMENTS FOR TREATING CANCER AMGEN INC. (US) 2006-06-08 WO disclosed