SCHEMBL5223225

SCHEMBL5223225

OCC(O)CNCc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1ccco1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
MAPT P10636 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.34
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CNKSR1 Q969H4 1/20 0.33
MAPK14 Q16539 2/20 0.33
GAK O14976 1/20 0.33
LCK P06239 1/20 0.33
PDGFRB P09619 1/20 0.33
MAPK9 P45984 1/20 0.33
MAPK10 P53779 1/20 0.33
EPHA5 P54756 1/20 0.33
MAPK11 Q15759 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224886 0.84 PTGS1 (0.37) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5228534 0.83 PTGS1 (0.36) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5230318 0.83 MAPT (0.36) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL13019206 0.82 PTGS1 (0.43) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5224632 0.82 ALDH1A1 (0.39) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5228370 0.81 ALDH1A1 (0.36) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5231186 0.80 SMN1; SMN2 (0.38) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5226789 0.78 ALDH1A1 (0.39) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5227606 0.78 TP53 (0.42) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5226514 0.78 PTGS1 (0.38) PTGS1NPSR1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed