SCHEMBL5226514

SCHEMBL5226514

Fc1ccc(-c2ccc(-n3ncc(CNC4CC4)c3-c3ccco3)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.38
NPSR1 Q6W5P4 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADORA2A P29274 2/20 0.35
ADORA1 P30542 1/20 0.35
NR3C1 P04150 1/20 0.34
HPGD P15428 2/20 0.34
CYP1A2 P05177 2/20 0.34
LMNA P02545 2/20 0.34
FLT3 P36888 1/20 0.34
ALOX12 P18054 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229163 0.96 USP2 (0.39) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5226654 0.86 BCHE (0.41) CYP3A4CYP2D6CYP2C19MAPTTP53
SCHEMBL5228622 0.85 MEN1 (0.46) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5224047 0.83 KDM4E (0.45) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL13019206 0.81 PTGS1 (0.43) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5231186 0.80 SMN1; SMN2 (0.38) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5224886 0.80 PTGS1 (0.37) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5224632 0.79 ALDH1A1 (0.39) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5228534 0.79 PTGS1 (0.36) PTGS1NPSR1CYP3A4CYP2D6CYP2C9
SCHEMBL5230318 0.78 MAPT (0.36) PTGS1NPSR1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed