SCHEMBL5223710

SCHEMBL5223710

CC(C)(C)N(C(=O)O)[C@@H](Cc1cc(F)cc(F)c1)[C@@H](O)CNCc1cccc(C(F)(F)F)c1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.57
BCHE P06276 4/20 0.50
CTSD P07339 10/20 0.46
BACE2 Q9Y5Z0 7/20 0.46
CTSB P07858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223705 1.00 BACE1 (0.57) BACE1BCHECTSDBACE2CTSB
SCHEMBL3016198 0.92 BACE1 (0.58) BACE1BCHECTSDBACE2
SCHEMBL3016194 0.92 BACE1 (0.58) BACE1BCHECTSDBACE2
SCHEMBL5375739 0.90 BACE1 (0.54) BACE1CTSDCTSB
SCHEMBL5219985 0.86 BACE1 (0.55) BACE1CTSDBACE2
SCHEMBL5219994 0.86 BACE1 (0.55) BACE1CTSDBACE2
SCHEMBL5224305 0.83 BACE1 (0.47) BACE1BCHECTSDBACE2
SCHEMBL5224294 0.83 BACE1 (0.47) BACE1BCHECTSDBACE2
SCHEMBL5383781 0.82 CTSD (0.54) BACE1CTSD
SCHEMBL5383784 0.82 CTSD (0.54) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed