SCHEMBL5224294

SCHEMBL5224294

CC(C)(C)N(C(=O)O)[C@@H](Cc1ccccc1)[C@H](O)CNCCc1cccc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.47
BCHE P06276 4/20 0.47
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
CTSD P07339 7/20 0.44
BACE2 Q9Y5Z0 7/20 0.44
CYP3A4 P08684 3/20 0.43
USP2 O75604 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
NR1I2 O75469 1/20 0.43
ADRB1 P08588 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
CHRM3 P20309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224305 1.00 BACE1 (0.47) BACE1BCHEKDM4EMEN1KMT2A
SCHEMBL3016198 0.90 BACE1 (0.58) BACE1BCHECTSDBACE2
SCHEMBL3016194 0.90 BACE1 (0.58) BACE1BCHECTSDBACE2
SCHEMBL5219646 0.88 ADRB3 (0.43) BACE1BCHEKDM4EMEN1KMT2A
SCHEMBL5219638 0.88 ADRB3 (0.43) BACE1BCHEKDM4EMEN1KMT2A
SCHEMBL5219515 0.86 SLC2A1 (0.46) MEN1KMT2AADRB1
SCHEMBL5219507 0.86 SLC2A1 (0.46) MEN1KMT2AADRB1
SCHEMBL5216394 0.84 OPRM1 (0.47) BACE1BCHEKDM4EMEN1KMT2A
SCHEMBL5216401 0.84 OPRM1 (0.47) BACE1BCHEKDM4EMEN1KMT2A
SCHEMBL5217761 0.83 PLAAT3 (0.43) MEN1KMT2AADRB1SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed