SCHEMBL5223855

SCHEMBL5223855

COc1ccc(-c2nn3ccccc3c2-c2ccnc(Cl)n2)cc1C1(F)C=CC=C(F)C1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 4/20 0.39
AURKA O14965 1/20 0.35
KDR P35968 1/20 0.35
AURKB Q96GD4 1/20 0.35
CDK19 Q9BWU1 1/20 0.35
MAPK9 P45984 7/20 0.33
MAPK8 P45983 6/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
EGFR P00533 4/20 0.33
RAF1 P04049 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
GSK3B P49841 1/20 0.33
MAPK14 Q16539 1/20 0.33
MAPK10 P53779 2/20 0.31
MAPK1 P28482 2/20 0.31
PDE4B Q07343 1/20 0.30
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226781 0.87 SLC2A1 (0.40) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL5223864 0.78 SLC2A1 (0.42) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3545328 0.77 MAPK1 (0.39) SLC2A1MAPK9EGFRRAF1ADORA3
SCHEMBL5223915 0.76 MAPK14 (0.34) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3441701 0.76 SLC2A1 (0.53) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3442348 0.74 SLC2A1 (0.41) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL5222821 0.74 KDR (0.48) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL4705773 0.73 SLC2A1 (0.35) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL5226655 0.72 SLC2A1 (0.40) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL12997420 0.71 GSK3B (0.50) MAPK9EGFRRAF1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828185-A2 2-PYRIMIDINYL PYRAZOLOPYRIDINE ERBB KINASE INHIBITORS SmithKline Beecham Corporation (US) 2007-09-05 EP disclosed
WO-2006068826-A2 2-PYRIMIDINYL PYRAZOLOPYRIDINE ERBB KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2006-06-29 WO disclosed