SCHEMBL5223864

SCHEMBL5223864

COc1ccc(-c2nn3ccccc3c2-c2ccnc(Cl)n2)cc1-c1ccc(F)c(C(N)=O)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 4/20 0.42
AURKA O14965 1/20 0.38
KDR P35968 1/20 0.38
AURKB Q96GD4 1/20 0.38
CDK19 Q9BWU1 1/20 0.38
SQOR Q9Y6N5 1/20 0.36
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
GSK3B P49841 2/20 0.35
EGFR P00533 1/20 0.35
RAF1 P04049 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
MAPK14 Q16539 1/20 0.35
BTK Q06187 3/20 0.34
MAPK8 P45983 3/20 0.34
MAPK9 P45984 3/20 0.34
JAK2 O60674 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225154 0.87 SLC2A1 (0.46) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3441701 0.81 SLC2A1 (0.53) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL5229307 0.81 SLC2A1 (0.44) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3545328 0.79 MAPK1 (0.39) SLC2A1GSK3BEGFRRAF1ADORA3
SCHEMBL5223855 0.78 SLC2A1 (0.39) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL4705773 0.77 SLC2A1 (0.35) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3442348 0.77 SLC2A1 (0.41) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3542508 0.76 GSK3B (0.46) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL5223920 0.76 MAPK14 (0.37) SLC2A1AURKAKDRAURKBCDK19
SCHEMBL3442312 0.75 SLC2A1 (0.55) SLC2A1AURKAKDRAURKBCDK19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828185-A2 2-PYRIMIDINYL PYRAZOLOPYRIDINE ERBB KINASE INHIBITORS SmithKline Beecham Corporation (US) 2007-09-05 EP disclosed
WO-2006068826-A2 2-PYRIMIDINYL PYRAZOLOPYRIDINE ERBB KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2006-06-29 WO disclosed