SCHEMBL5223874

SCHEMBL5223874

CC(C)(NC[C@@H](O)[C@@H](N)Cc1ccccc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR2B P41595 1/20 0.47
BACE1 P56817 6/20 0.46
CTSD P07339 7/20 0.46
BACE2 Q9Y5Z0 2/20 0.46
BCHE P06276 1/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
ACP3 P15309 1/20 0.42
F2 P00734 1/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
CSNK1E P49674 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224458 0.87 BACE1 (0.56) BACE1CTSDBCHEF2CSNK1E
SCHEMBL5222715 0.84 CTSD (0.58) CTSD
SCHEMBL3351844 0.81 BACE1 (0.54) BACE1CTSDF2ADRB1CSNK1E
SCHEMBL8276492 0.81 BACE1 (0.62) HTR2AHTR2CHTR2BBACE1CTSD
SCHEMBL161260 0.81 BACE1 (0.62) HTR2AHTR2CHTR2BBACE1CTSD
SCHEMBL3455222 0.81 BACE1 (0.62) HTR2AHTR2CHTR2BBACE1CTSD
SCHEMBL5385450 0.80 CTSD (0.44) HTR2AHTR2CHTR2BBACE1CTSD
Hydrochloric Acid SCHEMBL2499284 0.80 BACE1 (0.61) HTR2AHTR2CHTR2BBACE1CTSD
SCHEMBL5385448 0.79 CTSD (0.65) BACE1CTSDBACE2BCHE
SCHEMBL13315977 0.79 BACE1 (0.56) HTR2AHTR2CHTR2BBACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed