SCHEMBL5223970

SCHEMBL5223970

Fc1ccc(-c2ccc(-n3ncc(CN4CCN(CCN5CCCC5)CC4)c3-c3ccco3)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.40
SMO Q99835 2/20 0.40
MAPT P10636 1/20 0.38
KCNH2 Q12809 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
DRD2 P14416 4/20 0.38
DRD4 P21917 4/20 0.38
DRD3 P35462 4/20 0.38
PTGS1 P23219 1/20 0.37
MCHR1 Q99705 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
LMNA P02545 1/20 0.35
ADORA1 P30542 1/20 0.35
USP7 Q93009 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761009 0.91 SMO (0.43) ADORA2ASMOMAPTDRD2DRD4
SCHEMBL2761237 0.89 SMO (0.43) ADORA2ASMOMAPTDRD2DRD4
Hydrochloric Acid SCHEMBL1997589 0.88 SMO (0.42) ADORA2ASMOMAPTDRD2DRD4
SCHEMBL2761177 0.87 DRD4 (0.42) SMOMAPTDRD2DRD4DRD3
SCHEMBL2761137 0.86 SMO (0.41) SMOMAPTDRD2DRD4DRD3
SCHEMBL5228002 0.84 TSHR (0.39) SMOPTGS1MCHR1ALDH1A1SMN1; SMN2
SCHEMBL5224673 0.83 SMO (0.40) SMODRD2DRD4DRD3ALDH1A1
SCHEMBL5744201 0.81 CHKA (0.41) ADORA2ASMOMAPTDRD2DRD4
SCHEMBL5226032 0.81 SMO (0.39) SMODRD2DRD4DRD3PTGS1
SCHEMBL1995720 0.81 SMO (0.38) SMOMAPTDRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed