SCHEMBL5224322

SCHEMBL5224322

CN1CCN(Cc2cnn(-c3ccc(-c4ccc5c(c4)OCCO5)cc3)c2-n2cccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
LMNA P02545 6/20 0.51
USP2 O75604 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
TP53 P04637 1/20 0.51
TSHR P16473 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
POLB P06746 2/20 0.44
LCK P06239 1/20 0.42
MAP4K3 Q8IVH8 1/20 0.42
MAP4K1 Q92918 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
GAA P10253 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HTT P42858 1/20 0.41
MAPT P10636 2/20 0.40
INSR P06213 1/20 0.39
ALK Q9UM73 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224506 0.92 ALDH1A1 (0.51) ALDH1A1LMNAUSP2SMN1; SMN2TP53
SCHEMBL5229173 0.82 DRD4 (0.47) ALDH1A1LMNASMN1; SMN2TP53DRD4
SCHEMBL5230509 0.81 POLB (0.41) ALDH1A1SMN1; SMN2TP53TSHRPOLB
SCHEMBL2761292 0.78 LCK (0.41) ALDH1A1SMN1; SMN2POLBLCKMAP4K3
SCHEMBL5222920 0.76 ALDH1A1 (0.41) ALDH1A1LMNAUSP2SMN1; SMN2TP53
SCHEMBL2761054 0.76 MAPT (0.43) ALDH1A1LMNAUSP2SMN1; SMN2TP53
SCHEMBL5228465 0.74 SMO (0.46) ALDH1A1LMNAUSP2SMN1; SMN2MEN1
SCHEMBL5229195 0.74 POLB (0.40) ALDH1A1LMNAUSP2SMN1; SMN2TP53
SCHEMBL5907255 0.70 CYP2A13 (0.42) ALDH1A1LMNAUSP2SMN1; SMN2TP53
SCHEMBL5224327 0.70 KDM4E (0.36) ALDH1A1LMNAUSP2SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed