SCHEMBL5224749

SCHEMBL5224749

Cc1nnc(-c2ccc(-c3cc(NC(=O)Oc4ccoc4)ccc3C)cc2)o1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 20/20 0.53
LCK P06239 3/20 0.44
MAP2K1 Q02750 1/20 0.44
MAPK11 Q15759 2/20 0.43
HSPB1 P04792 1/20 0.43
CSF1R P07333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5122976 0.82 MAPK14 (0.62) MAPK14LCKMAP2K1MAPK11HSPB1
SCHEMBL14078280 0.74 MAPK14 (0.66) MAPK14LCKMAP2K1MAPK11HSPB1
SCHEMBL5220199 0.73 MAPK14 (0.50) MAPK14MAP2K1MAPK11
SCHEMBL5221091 0.73 MAPK14 (0.64) MAPK14LCKMAP2K1CSF1R
SCHEMBL5216405 0.72 MAPK14 (0.57) MAPK14MAP2K1MAPK11
SCHEMBL5113564 0.71 MAPK14 (0.61) MAPK14LCKMAP2K1MAPK11CSF1R
SCHEMBL4856439 0.69 MAPK14 (1.00) MAPK14LCKMAPK11
SCHEMBL14078304 0.69 MAPK14 (0.71) MAPK14LCKMAP2K1MAPK11CSF1R
SCHEMBL5122607 0.68 MAPK14 (0.60) MAPK14MAP2K1MAPK11
SCHEMBL4864546 0.68 MAPK14 (0.78) MAPK14LCKMAP2K1MAPK11CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499600-B1 HETEROARYL SUBSTITUTED BIPHENYL DERIVATIVES AS P38 KINASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-07-25 EP claimed