SCHEMBL5224931

SCHEMBL5224931

COc1ccc(-c2ccc(C(c3cn[nH]c3-c3ccccc3F)N3CCN(C)CC3)cc2)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHB4 P54760 1/20 0.41
KCNH2 Q12809 4/20 0.37
MAP4K1 Q92918 6/20 0.36
HTR2B P41595 2/20 0.36
HTR1A P08908 2/20 0.36
HTR7 P34969 1/20 0.36
HTR3A P46098 1/20 0.36
HTR6 P50406 1/20 0.36
AVPR2 P30518 1/20 0.35
OXTR P30559 1/20 0.35
AVPR1A P37288 1/20 0.35
CHRM2 P08172 2/20 0.34
ADRA2A P08913 2/20 0.34
CHRM1 P11229 2/20 0.34
DRD1 P21728 2/20 0.34
DRD3 P35462 2/20 0.34
SLC6A3 Q01959 2/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5907425 0.88 CHRM2 (0.43) KCNH2MAP4K1HTR2BHTR1AHTR7
SCHEMBL2761056 0.86 ALDH1A1 (0.43) MAP4K1HTR2BHTR1AHTR7HTR3A
SCHEMBL5228640 0.85 HTR2B (0.39) KCNH2MAP4K1HTR2BHTR1AHTR7
SCHEMBL5224222 0.84 MAP4K1 (0.39) KCNH2MAP4K1HTR2BHTR1AHTR7
SCHEMBL2761086 0.84 HTR2B (0.39) KCNH2MAP4K1HTR2BHTR1AHTR7
SCHEMBL7261976 0.83 HTR1A (0.42) KCNH2HTR2BHTR1AHTR7HTR3A
SCHEMBL5229983 0.83 ALDH1A1 (0.38) KCNH2MAP4K1HTR2BHTR1AHTR7
SCHEMBL5232124 0.83 HTR1A (0.38) KCNH2MAP4K1HTR2BHTR1AHTR7
SCHEMBL2761149 0.82 HTR2B (0.39) KCNH2MAP4K1HTR2BHTR1AHTR7
SCHEMBL5226498 0.81 HTR1A (0.38) KCNH2MAP4K1HTR2BHTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed