SCHEMBL5225271

SCHEMBL5225271

C1=CCCC(C2=COC=C(c3ccc(-n4ncc(CN5CCN(C6CCCC6)CC5)c4-c4ccco4)cc3)O2)=C1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.30
DRD2 P14416 1/20 0.30
HTR2A P28223 1/20 0.30
HRH1 P35367 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226178 0.90 AAK1 (0.31)
SCHEMBL5230515 0.89 DRD4 (0.30) DRD4DRD3
SCHEMBL5229202 0.89
SCHEMBL5227556 0.88
SCHEMBL5227647 0.86 F10 (0.33)
SCHEMBL5228480 0.85
SCHEMBL2901686 0.84 ALDH1A1 (0.36) ALDH1A1KDM4EDRD2HTR2AHRH1
SCHEMBL5227292 0.81
SCHEMBL5225931 0.81 TP53 (0.33) KDM4E
SCHEMBL5224958 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed