SCHEMBL5225931

SCHEMBL5225931

CC(C)(C)OC(=O)NC1CCN(Cc2cnn(-c3ccc(C4=COC=C(C5=CC=CCC5)O4)cc3)c2-c2ccco2)CC1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.33
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
KCNA3 P22001 1/20 0.33
AAK1 Q2M2I8 3/20 0.33
LMNA P02545 3/20 0.33
AKT1 P31749 1/20 0.33
F2 P00734 1/20 0.32
F10 P00742 1/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32
MAPT P10636 1/20 0.32
THRB P10828 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226178 0.85 AAK1 (0.31) AAK1
SCHEMBL5230515 0.83 DRD4 (0.30)
SCHEMBL5225271 0.81 DRD4 (0.34) KDM4E
SCHEMBL5225926 0.78 MCHR1 (0.41) TP53AAK1LMNAMAPTTHRB
SCHEMBL2901963 0.74 ABCB1 (0.36) MAPTKDM4E
SCHEMBL5907258 0.69 CYP2A13 (0.37) F2F10
SCHEMBL5224327 0.68 KDM4E (0.36) TP53LMNAMAPTKDM4E
SCHEMBL5224513 0.68 KDM4E (0.36) TP53LMNAMAPTKDM4E
SCHEMBL2908338 0.68 ALDH1A1 (0.37) LMNAF2F10MAPTKDM4E
SCHEMBL2904995 0.67 ALDH1A1 (0.38) PARP1PARP2LMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed