SCHEMBL5225340

SCHEMBL5225340

COc1cccc(CC(C)(C)NC[C@@H](O)[C@@H](N)Cc2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASR P41180 9/20 0.52
TAAR1 Q96RJ0 2/20 0.47
ADRB2 P07550 1/20 0.46
ADRB1 P08588 1/20 0.46
F2 P00734 1/20 0.45
CTSD P07339 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5222715 0.85 CTSD (0.58) CTSD
SCHEMBL5217674 0.85 CSNK1E (0.49) CASRADRB2F2
SCHEMBL5383193 0.83 CASR (0.46) CASRADRB2ADRB1F2
SCHEMBL3353932 0.82 BCHE (0.52) TAAR1ADRB2ADRB1F2CTSD
Hydrochloric Acid SCHEMBL5222886 0.82 CASR (0.45) CASRADRB2ADRB1F2
SCHEMBL165644 0.82 BCHE (0.61) CTSD
SCHEMBL4214871 0.82 BCHE (0.61) CTSD
Hydrochloric Acid SCHEMBL5225498 0.81 BCHE (0.51) TAAR1ADRB2ADRB1F2CTSD
Hydrochloric Acid SCHEMBL5348922 0.81 BCHE (0.60) CTSD
Hydrochloric Acid SCHEMBL6110582 0.81 BCHE (0.60) CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed