SCHEMBL5225757

SCHEMBL5225757

CN(C)CCN1C(=O)[C][C@H](c2cccc(Cl)c2)Sc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 0.50
ICAM1 P05362 1/20 0.50
ITGAL P20701 1/20 0.50
KDM1A O60341 3/20 0.44
CACNA1S Q13698 4/20 0.44
CACNA1C Q13936 3/20 0.44
LMNA P02545 4/20 0.43
CYP3A4 P08684 4/20 0.43
KCNH2 Q12809 4/20 0.43
TP53 P04637 4/20 0.43
MAPT P10636 3/20 0.43
CYP1A2 P05177 3/20 0.43
HTR1A P08908 3/20 0.43
CYP2D6 P10635 3/20 0.43
DRD2 P14416 3/20 0.43
CYP2C19 P33261 3/20 0.43
ABCB11 O95342 3/20 0.43
SLC22A1 O15245 3/20 0.43
HRH2 P25021 3/20 0.43
ADRA1A P35348 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3343427 0.82 GSK3B (0.43) TP53MAPTSMN1; SMN2RAB9ASLC6A3
SCHEMBL11435169 0.80 CACNA1S (0.65) KDM1ACACNA1SCACNA1CLMNACYP3A4
SCHEMBL5225360 0.78 CACNA1S (0.55) ITGB2ICAM1ITGALKDM1ACACNA1S
SCHEMBL10809571 0.71 ITGB2 (0.53) ITGB2ICAM1ITGALKDM1ACACNA1S
SCHEMBL3346744 0.69 OPRK1 (0.40) ITGB2ICAM1ITGALKDM1ACACNA1S
Hydrochloric Acid SCHEMBL9505100 0.69 ITGB2 (0.50) ITGB2ICAM1ITGALKDM1ACACNA1S
Thiazesim SCHEMBL30263577 0.69 GSK3B (0.65) KDM1ACACNA1STP53MAPTSMN1; SMN2
Thiazesim SCHEMBL49862 0.69 GSK3B (0.65) KDM1ACACNA1STP53MAPTSMN1; SMN2
SCHEMBL10808149 0.68 ITGB2 (0.55) ITGB2ICAM1ITGALKDM1ACACNA1S
SCHEMBL10538420 0.68 CACNA1S (0.60) ITGB2ICAM1ITGALKDM1ACACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1845089-A1 Novel lactams and uses thereof AstraZeneca AB (SE) 2007-10-17 EP disclosed