SCHEMBL5226079

SCHEMBL5226079

COc1ccc(NC(=O)c2ccccc2NC(=O)c2ccc(CC(C)O)cc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.73
NPC1 O15118 6/20 0.65
RAB9A P51151 5/20 0.65
POLB P06746 2/20 0.65
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65
PPARD Q03181 1/20 0.60
TDP1 Q9NUW8 2/20 0.59
PKM P14618 1/20 0.59
RXFP1 Q9HBX9 2/20 0.56
F10 P00742 4/20 0.56
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 1/20 0.55
HPGD P15428 1/20 0.55
TP53 P04637 1/20 0.54
ALOX15 P16050 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HDAC1 Q13547 1/20 0.53
NR1H4 Q96RI1 1/20 0.53
MAPT P10636 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227999 0.85 NPC1 (0.69) ABCG2NPC1RAB9APOLBMEN1
SCHEMBL5223096 0.84 RAB9A (0.71) ABCG2NPC1RAB9APOLBMEN1
SCHEMBL5226517 0.83 NPC1 (0.76) ABCG2NPC1RAB9APOLBMEN1
SCHEMBL5223218 0.81 NR1H4 (0.73) ABCG2NPC1RAB9APOLBMEN1
SCHEMBL20715740 0.80 NPC1 (0.71) ABCG2NPC1RAB9AMEN1KMT2A
SCHEMBL5225155 0.80 NPC1 (0.71) ABCG2NPC1RAB9APOLBMEN1
SCHEMBL5226076 0.80 NPC1 (0.71) ABCG2NPC1RAB9APOLBMEN1
SCHEMBL5188942 0.79 NPC1 (1.00) ABCG2NPC1RAB9APOLBMEN1
SCHEMBL1689196 0.77 HDAC1 (0.78) ABCG2F10HDAC1
SCHEMBL14855681 0.77 F10 (0.72) ABCG2NPC1RAB9APOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1014962-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2007-06-27 EP disclosed
EP-1014962-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1999000121-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1999-01-07 WO disclosed