SCHEMBL5226654

SCHEMBL5226654

Fc1ccc(CCN2CCC(NCc3cnn(-c4ccc(-c5ccc(F)cc5)cc4)c3-c3ccco3)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.41
ACHE P22303 4/20 0.41
BACE1 P56817 4/20 0.41
OPRM1 P35372 2/20 0.36
EED O75530 2/20 0.36
SSTR5 P35346 2/20 0.36
KCNH2 Q12809 2/20 0.34
NR4A2 P43354 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
EHMT2 Q96KQ7 1/20 0.34
DNMT3A Q9Y6K1 1/20 0.34
CYP2D6 P10635 2/20 0.33
CHRM1 P11229 2/20 0.33
DRD2 P14416 2/20 0.33
DRD4 P21917 2/20 0.33
HTR2A P28223 2/20 0.33
MEN1 O00255 1/20 0.33
MLNR O43193 1/20 0.33
CACNA1F O60840 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226514 0.86 PTGS1 (0.38) CYP2D6USP2LMNATP53CYP1A2
SCHEMBL5229163 0.84 USP2 (0.39) HRH3CYP2D6USP2LMNATP53
SCHEMBL5228622 0.79 MEN1 (0.46) CYP2D6CHRM1MEN1TP53CHRM2
SCHEMBL5225875 0.75 CYP2D6 (0.36) CYP2D6DRD2DRD4TP53CYP3A4
SCHEMBL5226789 0.74 ALDH1A1 (0.39) CYP2D6MEN1LMNATP53CYP3A4
SCHEMBL5222786 0.74 GRM2 (0.38) KCNH2HRH3CYP2D6TP53HRH1
SCHEMBL5224047 0.74 KDM4E (0.45) CYP2D6LMNATP53CYP3A4MAPT
SCHEMBL2761009 0.74 SMO (0.43) DRD2DRD4LMNATP53MAPT
SCHEMBL5228002 0.73 TSHR (0.39) ACHETP53HTR2CHTTKMT2A
SCHEMBL5223970 0.73 ADORA2A (0.40) KCNH2HRH3DRD2DRD4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed