SCHEMBL5226760

SCHEMBL5226760

[CH2]CCC(C#N)(c1ccccc1)C(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EBP Q15125 2/20 0.56
SIGMAR1 Q99720 2/20 0.56
CYP3A4 P08684 7/20 0.42
CYP2D6 P10635 4/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
DRD2 P14416 3/20 0.41
OPRM1 P35372 3/20 0.41
DRD3 P35462 3/20 0.41
DRD4 P21917 2/20 0.41
CYP2C19 P33261 3/20 0.38
ABCB1 P08183 5/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ATM Q13315 1/20 0.35
CHRM2 P08172 2/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CYP3A5 P20815 1/20 0.34
RIPK1 Q13546 1/20 0.34
KCNA3 P22001 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7753625 0.86 EBP (0.56) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL7310080 0.81 EBP (0.59) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL5236598 0.81 EBP (0.59) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL5242023 0.81 EBP (0.59) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL8751165 0.81 EBP (0.59) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL7310837 0.81 EBP (0.52) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL5237762 0.81 EBP (0.59) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL5752959 0.80 EBP (0.51) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL5751980 0.80 EBP (0.51) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1
SCHEMBL7310593 0.80 EBP (0.51) EBPSIGMAR1CYP3A4CYP2D6L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1818326-A1 Nitrogen-containing heterocyclic compounds and pharmaceutical composition containing the compounds Eisai R&D Management Co., Ltd. (JP) 2007-08-15 EP disclosed
EP-1254895-B1 NITROGENOUS CYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME EISAI R&D MAN CO LTD (JP) 2007-05-23 EP disclosed